TABLETS
Are Unit dosage form, tamperproof solid dosage form.
Manufacture of Granulations
Direct
Compression
e.g. NaCl, KBr etc.
Compression granulation Wet granulation
Direct compression: Some crystalline substances which can be compressed directly. A directly compressible
diluents added e.g. microcrystalline cellulose.
Disadvantages:
9 Differences in particle size & bulk density between drug & diluents leads to stratification within granulation
resulting in poor content of uniformity of drug in compressed tablet.
9 In direct compression diluents may interact with the drug e.g. Milard’s reaction that is yellow discolouration
between amine groups and hydrous lactose.
9 Because of dry nature of direct compression a static charge develops which may prevent uniform distribution of
drug in the granulation.
9 The maximum percentage of non compressible content in direct compression can be upto 30%.
Compression granulations: Used when drug is sensitive to heat, moisture (wet granulations) e.g. vitamins, aspirin
etc.
Powder blend slugs
՜
Screened or milled to produce granular form
Equipments:
1. Roller Compactor
2. Chilsonator
3. Hut’s compactor
Are Unit dosage form, tamperproof solid dosage form.
Manufacture of Granulations
Direct
Compression
e.g. NaCl, KBr etc.
Compression granulation Wet granulation
Direct compression: Some crystalline substances which can be compressed directly. A directly compressible
diluents added e.g. microcrystalline cellulose.
Disadvantages:
9 Differences in particle size & bulk density between drug & diluents leads to stratification within granulation
resulting in poor content of uniformity of drug in compressed tablet.
9 In direct compression diluents may interact with the drug e.g. Milard’s reaction that is yellow discolouration
between amine groups and hydrous lactose.
9 Because of dry nature of direct compression a static charge develops which may prevent uniform distribution of
drug in the granulation.
9 The maximum percentage of non compressible content in direct compression can be upto 30%.
Compression granulations: Used when drug is sensitive to heat, moisture (wet granulations) e.g. vitamins, aspirin
etc.
Powder blend slugs
՜
Screened or milled to produce granular form
Equipments:
1. Roller Compactor
2. Chilsonator
3. Hut’s compactor
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